Search results for "acid catalysi"

showing 10 items of 58 documents

ChemInform Abstract: Influence of Reactant Polarity on the Course of the Inverse-Electron-Demand Diels-Alder Reaction. A DFT Study of Regio- and Ster…

2010

The molecular mechanisms for the inverse-electron-demand Diels−Alder reactions between nitroethene and three substituted ethenes (propene, methyl vinyl ether, and dimethylvinylamine) to give the corresponding nitroso cycloadducts have been characterized with density functional theory methods using the B3LYP/6-31G* calculational level. On the basis of stability arguments and molecular orbital analysis relative rates, regioselectivity, and stereoselectivity, the presence of Lewis acid catalyst modeled by the BH3 system and the inclusion of solvent effects as a function of the nature of substituent in the dienophile fragment are analyzed and discussed. The ortho attack mode presents transition…

chemistry.chemical_compoundchemistrySubstituentRegioselectivityStereoselectivityGeneral MedicineMethyl vinyl etherNitrosoSolvent effectsInverse electron-demand Diels–Alder reactionMedicinal chemistryLewis acid catalysisChemInform
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On the Rearrangement in Dioxane/Water of (Z)-Arylhydrazones of 5-Amino-3-benzoyl-1,2,4-oxadiazole into (2-Aryl-5-phenyl-2H-1,2,3-triazol-4-yl)ureas: …

2006

We have recently evidenced an interesting differential behavior in the reactivity in dioxane/water between the (Z)-2,4-dinitrophenylhydrazone (1a) and the (Z)-phenylhydrazone (1b) of 5-amino-3-benzoyl-1,2,4- oxadiazole. The former rearranges into the relevant triazole 2a only at pS+ > 4.5 while undergoing hydrolysis at high proton concentration (pS+ < 3.5); on the contrary, the latter rearranges into 2b in the whole pS+ range examined (0.1 e pS+ e 14.9). Thus, for a deeper understanding of these differences we have now collected kinetic data on the rearrangement in dioxane/water of a series of 3- or 4-substituted (Z)-phenylhydrazones (1c-l) of 5-amino-3-benzoyl-1,2,4-oxadiazole in a wide ra…

OxadiazolesMolecular StructureStereochemistryArylOrganic ChemistryHydrazonesTriazoleSubstituentWaterOxadiazolemononuclear rearrangement of heterocycles acid catalysis base catalysisTriazolesChemical synthesisMedicinal chemistryCatalysisDioxanesKineticschemistry.chemical_compoundAcid catalysischemistryThermodynamicsAmine gas treatingReactivity (chemistry)
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Exploring the potential of some yeast strains in the stereoselective synthesis of aldol reaction products and its reduced 1,3-dialcohol derivatives

2013

Abstract The behavior of two yeast strains has been studied under different conditions. Both microorganims catalyzed the aldol reaction between activated aldehydes and acetone when a large amount of the latter was present in the reaction medium producing, with moderate stereoselectivity, the aldol product with the R configuration. No reduction of any of the products present in the medium was detected. On the other hand, the carbonyl group of the racemic aldol was reduced to produce chiral 1,3-dialcohol derivatives when water was employed as the only solvent. In this case, the resolution of the racemic starting material was also possible with one of the biocatalysts, and the aldol was recove…

ChemistryProcess Chemistry and TechnologyCarbonyl reductionEnantioselective synthesisBioengineeringBiochemistryCatalysisLewis acid catalysisStereocenterAldol reactionBiocatalysisOrganic chemistryAldol condensationStereoselectivityJournal of Molecular Catalysis B: Enzymatic
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Using theozymes for designing transition-state analogs for the intramolecular aldol reaction of δ-diketones

2001

Two theozymes for the intramolecular aldol reaction of δ-diketones have been studied using ab initio methods. The presence of both acid/base residues favors several steps of the aldol reaction. The appropriate positioning of these residues can accelerate one of two diastereromeric reaction pathways, the catalyzed aldol reaction being highly stereoselective. Analysis of the geometrical parameters, charge distribution, and the shape of molecular electrostatic potential for the corresponding acid/base catalyzed transition structure allows us to design adequate transition-state analogs to favor a reactive channel of this intramolecular aldol reaction. © 2001 John Wiley & Sons, Inc. Int J Quant …

ChemistryStereochemistryorganic chemicalsAb initioCondensed Matter PhysicsAtomic and Molecular Physics and OpticsCatalysisLewis acid catalysisAldol reactionTransition state analogAb initio quantum chemistry methodsIntramolecular forcepolycyclic compoundsStereoselectivityPhysical and Theoretical ChemistryInternational Journal of Quantum Chemistry
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Zur protonenkatalysierten Xanthenylierung von Tryptamin, Nω-Acetyltryptamin und Gramin: Ein Beitrag zur Konstitutionsaufklärung in der Indol-Analytik

1988

Acid catalysisAcetic acidchemistry.chemical_compoundBicyclic moleculeChemistryDrug DiscoveryPharmaceutical ScienceAmine gas treatingAlcoholMedicinal chemistryArchiv der Pharmazie
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Can Macroscopic Parameters, Such as Conversion and Selectivity, Distinguish between Different Cracking Mechanisms on Acid Catalysts?

1997

n-heptane cracking has been carried out for very short time periods on an established reaction mechanism which includes the following group of stream reactions on different zeolites: Initiation reactions (protolytic cracking), charge isomerization, chain isomerization, hydride transfer, β-scission–alkylation, desorption–adsorption, and hydrogen transfer–cyclization. It has been observed that a given experimental distribution of products can be explained by more than just one reaction scheme. This does not allow one to clearly distinguish the fraction of reactant which disappears via monomolecular initiation reactions with respect to bimolecular hydride transfer reactions.

Acid catalysisReaction mechanismCrackingHydrogenChemistryHydridechemistry.chemical_elementPhysical and Theoretical ChemistryPhotochemistryFluid catalytic crackingIsomerizationCatalysisCatalysisJournal of Catalysis
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The Reactions of Electron-Rich Heterocycles with Derivatives of Orthocarboxylic Acids; VIII. Proton Acid-Catalyzed Acylation of Indoles by 2-Alkoxy-1…

1987

In acid-catalyzed reactions with 3-unsubstituted indoles 1, 2-alkoxy-1,3-dioxolanes 2a-c behave as acyl equivalents. Depending on the substitution patterns of the reaction partners, the 1,3-dioxolanium ions 3a-c, generated in situ from the cyclic ortho esters by the action of sulfosalicylic acid, react to form tris-(3-indolyl)alkanes 6 and 9, bis-(3-indolyl)ethenes 7, or 3-benzoylindoles 8. Analogous reactivity was observed with related acyclic ortho esters. Reaktionen elektronenreicher Heterocyclen mit Orthocarbonsaure-Derivaten; VIII. Protonsaurekatalysierte Acylierung von Indolen mit 2-Alkoxy-1,3-dioxolanen 2-Alkoxy-1,3-dioxolane 2a-c reagieren als Acylaquivalente mit 3-unsubstituierten …

Indole testSulfosalicylic acidBicyclic moleculeStereochemistryPharmaceutical ScienceMedicinal chemistryAcylationchemistry.chemical_compoundAcid catalysischemistryDrug DiscoveryAlkoxy groupReactivity (chemistry)OrthoesterArchiv der Pharmazie
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Proton Acid-Catalysed Transformations of Estrogen Derivatives: New Results and Some Mechanistic Aspects of theKober Colour Reaction

1994

The 3-O-methylated estrogen derivatives 1a-d and α-estradiol (1e) underwent sulfuric acid-catalysed transformations to furnish the steroids 2–6. The processes involved in the reaction sequence are regioselective sulfonation and, above all, the Wagner-Meerwein rearrangement of the methyl group at C-13. With the objective of obtaining further information on the course of the Kober colour reaction of estrogens, some UV/VIS and ESR spectroscopic investigations were also carried out. Protonenkatalysierte Transformationen von Estrogen-Derivaten: Neue Ergebnisse und einige mechanistische Aspekte der Kober-Farbreaktion Die O-methylierten Estrogenderivate 1a-d und α-Estradiol (1e) reagieren in Schwe…

Wagner–Meerwein rearrangementStereochemistrymedicine.drug_classColor reactionPharmaceutical ScienceRegioselectivityEtherchemistry.chemical_compoundAcid catalysischemistryEstrogenDrug DiscoverymedicinePhenolsMethyl groupArchiv der Pharmazie
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The Pd3(dppm)3(CO)2+ Cluster: An Efficient Electrochemically Assisted Lewis Acid Catalyst for the Fluorination and Alcoholysis of Acyl Chlorides.

2002

The dicationic palladium cluster Pd3(dppm)3(CO)2+ (dppm = bis(diphenylphosphino)methane) reacts with acid chlorides RCOCl (R = n-C6H13, t-Bu, Ph) to afford quantitatively the chloride adduct Pd3(dppm)3(CO)(Cl)+ and the acyl cation RCO+ as the organic counterpart. The dicationic reactive cluster can be reformed by electrolyzing the chloride complex with a copper anode leaving CuCl as a byproduct. The combination of these two reactions provides an electrocatalytic way to form the acylium from the acid chloride. Indeed, in CH2Cl2, 0.2 M NBu4PF6, or NBu4BF4, the electrolysis of the acid chloride in the presence of a catalytic amount of the cluster (1%) gives in good yields the acid fluoride RCO…

ElectrolysisSupporting electrolyteOrganic ChemistryInorganic chemistrychemistry.chemical_elementGeneral MedicineElectrochemistryMedicinal chemistryChlorideAdductlaw.inventionLewis acid catalysisCatalysischemistry.chemical_compoundAcyl chloridechemistryNucleophilelawmedicineLewis acids and basesPalladiummedicine.drugChemInform
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2H -[1,3]Oxazino[3,2-α]indolin-4(3H )-ones: A Class Of Polyheterocyclic Indole-Based Compounds

2018

Indole testClass (set theory)Acid catalysis010405 organic chemistryStereochemistryChemistryOrganic ChemistryPhysical and Theoretical Chemistry010402 general chemistry01 natural sciences0104 chemical sciencesEuropean Journal of Organic Chemistry
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